Academic Bibliography

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Structure-activity relationship in monosaccharide-based Toll-like receptor 4 (TLR4) antagonists

Fabio A Facchini, Lenny Zaffaroni, Alberto Minotti, Silvia Rapisarda, Valentina Calabrese, Matilde Forcella, Paola Fusi, Cristina Airoldi, Carlotta Ciaramelli, Jean-Marc Billod, et al.

(2018) JOURNAL OF MEDICINAL CHEMISTRY. 61(7). p.2895-2909
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Medicinal chemistry and use of myosin II inhibitor (S)-blebbistatin and its derivatives

Bart Roman (UGent), Sigrid Verhasselt (UGent) and Christian Stevens (UGent)

(2018) JOURNAL OF MEDICINAL CHEMISTRY.
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Tozasertib analogues as inhibitors of necroptotic cell death

Sam Hofmans, Lars Devisscher, Sofie Martens (UGent), Dries Van Rompaey, Kenneth Goossens, Tatyana Divert (UGent), Wim Nerinckx (UGent), Nozomi Takahashi (UGent), Hans De Winter, Pieter Van der Veken, et al.

(2018) JOURNAL OF MEDICINAL CHEMISTRY. 61(5). p.1895-1920
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Design and syntheses of highly potent teixobactin analogues against Staphylococcus aureus, methicillin-resistant Staphylococcus aureus (MRSA), vancomycin-resistant Enterococci (VRE) in vitro and in vivo

Anish Parmar, Rajamani Lakshminarayanan, Abhishek Iyer (UGent), Venkatesh Mayandi, Eunice Tze Leng Goh, Daniel G Lloyd, Madhavi Latha S Chalasani, Navin Kumar Verma, Stephen H Prior, Roger W Beuerman, et al.

(2018) JOURNAL OF MEDICINAL CHEMISTRY. 61(5). p.2009-2017
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Determination of in vitro and in silico indexes for the modeling of blood-brain barrier partitioning of drugs via micellar and immobilized artificial membrane liquid chromatography

Giacomo Russo (UGent), Lucia Grumetto, Roman Szucs (UGent), Francesco Barbato and Frederic Lynen (UGent)

(2017) JOURNAL OF MEDICINAL CHEMISTRY. 60(9). p.3739-3754
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Novel ferroptosis inhibitors with improved potency and ADME properties

Sam Hofmans, Tom Vanden Berghe (UGent), Lars Devisscher, Behrouz Hassannia (UGent), Sophie Lyssens, Jurgen Joossens, Pieter Van Der Veken, Peter Vandenabeele (UGent) and Koen Augustyns

(2016) JOURNAL OF MEDICINAL CHEMISTRY. 59(5). p.2041-2053
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Synthesis and bioactivity of β-substituted fosmidomycin analogues targeting 1-deoxy-D-xylulose-5-phosphate reductoisomerase

René Chofor, Sanjeewani Sooriyaarachchi, Martijn Risseeuw (UGent), Terese Bergfors, Jenny Pouyez, Chinchu Johny, Amanda Haymond, Annelien Everaert, Cynthia S Dowd, Louis Maes, et al.

(2015) JOURNAL OF MEDICINAL CHEMISTRY. 58(7). p.2988-3001
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Structural investigation of B-Raf paradox breaker and inducer inhibitors

Rohit Arora, Michela Di Michele, Elisabeth Stes, Elien Vandermarliere (UGent), Lennart Martens (UGent), Kris Gevaert (UGent), Erika Van Heerde, Joannes TM Linders, Dirk Brehmer, Edgar Jacoby, et al.

(2015) JOURNAL OF MEDICINAL CHEMISTRY. 58(4). p.1818-1831
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1,2,3,4,8,9,10,11-Octahydrobenzo[j]phenanthridine-7,12-diones as new leads against Mycobacterium tuberculosis

Davie Cappoen, Pieter Claes (UGent), Jan Jacobs (UGent), Roel Anthonissen, Vanessa Mathys, Luc Verschaeve, Kris Huygen and Norbert De Kimpe (UGent)

(2014) JOURNAL OF MEDICINAL CHEMISTRY. 57(7). p.2895-2907
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Development of αGlcN(1 <-> 1)αMan-based Lipid A mimetics as a novel class of potent Toll-like Receptor 4 agonists

Florian Adanitsch, Simon Ittig, Johannes Stöckl, Alja Oblak, Mira Haegman (UGent), Roman Jerala, Rudi Beyaert (UGent), Paul Kosma and Alla Zamyatina

(2014) JOURNAL OF MEDICINAL CHEMISTRY. 57(19). p.8056-8071

Academic Bibliography

Biblio has been updated

Structure-activity relationship in monosaccharide-based Toll-like receptor 4 (TLR4) antagonists

Medicinal chemistry and use of myosin II inhibitor (S)-blebbistatin and its derivatives

Tozasertib analogues as inhibitors of necroptotic cell death

Design and syntheses of highly potent teixobactin analogues against Staphylococcus aureus, methicillin-resistant Staphylococcus aureus (MRSA), vancomycin-resistant Enterococci (VRE) in vitro and in vivo

Determination of in vitro and in silico indexes for the modeling of blood-brain barrier partitioning of drugs via micellar and immobilized artificial membrane liquid chromatography

Novel ferroptosis inhibitors with improved potency and ADME properties

Synthesis and bioactivity of β-substituted fosmidomycin analogues targeting 1-deoxy-D-xylulose-5-phosphate reductoisomerase

Structural investigation of B-Raf paradox breaker and inducer inhibitors

1,2,3,4,8,9,10,11-Octahydrobenzo[j]phenanthridine-7,12-diones as new leads against Mycobacterium tuberculosis

Development of αGlcN(1 <-> 1)αMan-based Lipid A mimetics as a novel class of potent Toll-like Receptor 4 agonists

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