Ghent University Academic Bibliography

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journalArticle
A1
open access

Structure-activity relationship in monosaccharide-based Toll-like receptor 4 (TLR4) antagonists

Fabio A Facchini, Lenny Zaffaroni, Alberto Minotti, Silvia Rapisarda, Valentina Calabrese, Matilde Forcella, Paola Fusi, Cristina Airoldi, Carlotta Ciaramelli, Jean-Marc Billod, et al.

(2018) JOURNAL OF MEDICINAL CHEMISTRY. 61(7). p.2895-2909

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Structure guided lead generation toward nonchiral M. tuberculosis thymidylate kinase inhibitors

Lijun Song (UGent) , Romain Merceron (UGent) , Begoña Gracia, Ainhoa Lucía Quintana, Martijn Risseeuw (UGent) , Fabian Hulpia (UGent) , Paul Cos, José A Aínsa, Hélène Munier-Lehmann, Savvas Savvides (UGent) , et al.

(2018) JOURNAL OF MEDICINAL CHEMISTRY. 61(7). p.2753-2775

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Discovery of novel 7-aryl 7-deazapurine 3'-deoxy-ribofuranosyl nucleosides with potent activity against Trypanosoma cruzi

Fabian Hulpia (UGent) , Kristof Van Hecke (UGent) , Cristiane Franca da Silva, Denise da Gama Jaen Batista, Louis Maes, Guy Caljon, Maria de Nazare C Soeiro and Serge Van Calenbergh (UGent)

(2018) JOURNAL OF MEDICINAL CHEMISTRY. 61(20). p.9287-9300

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Synthesis toward bivalent ligands for the dopamine D2 and metabotropic glutamate 5 receptors

Mingcheng Qian (UGent) , Elise Wouters (UGent) , James AR Dalton, Martijn Risseeuw (UGent) , René Crans (UGent) , Christophe Stove (UGent) , Jesús Giraldo, Kathleen Van Craenenbroeck (UGent) and Serge Van Calenbergh (UGent)

(2018) JOURNAL OF MEDICINAL CHEMISTRY. 61(18). p.8212-8225

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Tozasertib analogues as inhibitors of necroptotic cell death

Sam Hofmans, Lars Devisscher, Sofie Martens (UGent) , Dries Van Rompaey, Kenneth Goossens, Tatyana Divert (UGent) , Wim Nerinckx (UGent) , Nozomi Takahashi (UGent) , Hans De Winter, Pieter Van der Veken, et al.

(2018) JOURNAL OF MEDICINAL CHEMISTRY. 61(5). p.1895-1920

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Biodegradable amphipathic peptide hydrogels as extended-release system for opioid peptides

Charlotte Martin, Maria Dumitrascuta, Morgane Mannes, Aquilino Lantero, Dominik Bucher, Katja Walker, Yannick Van Wanseele, Edith Oyen, Sophie Hernot, Ann Van Eeckhaut, et al.

(2018) JOURNAL OF MEDICINAL CHEMISTRY. 61(21). p.9784-9789

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Design and syntheses of highly potent teixobactin analogues against Staphylococcus aureus, methicillin-resistant Staphylococcus aureus (MRSA), vancomycin-resistant Enterococci (VRE) in vitro and in vivo

Anish Parmar, Rajamani Lakshminarayanan, Abhishek Iyer (UGent) , Venkatesh Mayandi, Eunice Tze Leng Goh, Daniel G Lloyd, Madhavi Latha S Chalasani, Navin Kumar Verma, Stephen H Prior, Roger W Beuerman, et al.

(2018) JOURNAL OF MEDICINAL CHEMISTRY. 61(5). p.2009-2017

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Discovery of novel, drug-like ferroptosis inhibitors with in vivo efficacy

Lars Devisscher, Samya Van Coillie (UGent) , Sam Hofmans, Dries Van Rompaey, Kenneth Goossens, Eline Meul (UGent) , Louis Maes, Hans De Winter, Pieter Van Der Veken, Peter Vandenabeele (UGent) , et al.

(2018) JOURNAL OF MEDICINAL CHEMISTRY. 61(22). p.10126-10140

Mark

journalArticle
A1
open access

Determination of in vitro and in silico indexes for the modeling of blood-brain barrier partitioning of drugs via micellar and immobilized artificial membrane liquid chromatography

Giacomo Russo (UGent) , Lucia Grumetto, Roman Szucs (UGent) , Francesco Barbato and Frederic Lynen (UGent)

(2017) JOURNAL OF MEDICINAL CHEMISTRY. 60(9). p.3739-3754

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Novel ferroptosis inhibitors with improved potency and ADME properties

Sam Hofmans, Tom Vanden Berghe (UGent) , Lars Devisscher, Behrouz Hassannia (UGent) , Sophie Lyssens, Jurgen Joossens, Pieter Van Der Veken, Peter Vandenabeele (UGent) and Koen Augustyns

(2016) JOURNAL OF MEDICINAL CHEMISTRY. 59(5). p.2041-2053

Academic Bibliography

Structure-activity relationship in monosaccharide-based Toll-like receptor 4 (TLR4) antagonists

Structure guided lead generation toward nonchiral M. tuberculosis thymidylate kinase inhibitors

Discovery of novel 7-aryl 7-deazapurine 3'-deoxy-ribofuranosyl nucleosides with potent activity against Trypanosoma cruzi

Synthesis toward bivalent ligands for the dopamine D2 and metabotropic glutamate 5 receptors

Tozasertib analogues as inhibitors of necroptotic cell death

Biodegradable amphipathic peptide hydrogels as extended-release system for opioid peptides

Design and syntheses of highly potent teixobactin analogues against Staphylococcus aureus, methicillin-resistant Staphylococcus aureus (MRSA), vancomycin-resistant Enterococci (VRE) in vitro and in vivo

Discovery of novel, drug-like ferroptosis inhibitors with in vivo efficacy

Determination of in vitro and in silico indexes for the modeling of blood-brain barrier partitioning of drugs via micellar and immobilized artificial membrane liquid chromatography

Novel ferroptosis inhibitors with improved potency and ADME properties

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