Ghent University Academic Bibliography

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Dual-acting small molecules : subtype-selective cannabinoid receptor 2 agonist/butyrylcholinesterase inhibitor hybrids show neuroprotection in an Alzheimer's disease mouse model

Philipp Spatz, Sophie A. M. Steinmüller, Anna Tutov, Eleonora Poeta, Axelle Morilleau, Allison Carles, Marie Deventer (UGent) , Julian Hofmann, Christophe Stove (UGent) , Barbara Monti, et al.

(2023) JOURNAL OF MEDICINAL CHEMISTRY. 66(9). p.6414-6435
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The zinc-binding group effect : lessons from non-hydroxamic acid vorinostat analogs

Silke Geurs (UGent) , Dorien Clarisse (UGent) , Karolien De Bosscher (UGent) and Matthias D'hooghe (UGent)

(2023) JOURNAL OF MEDICINAL CHEMISTRY. 66(12). p.7698-7729
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Discovery of ss-arrestin-biased 25CN-NBOH-derived 5-HT2A receptor agonists

Christian B. M. Poulie, Eline Pottie (UGent) , Icaro A. Simon, Kasper Harpsoe, Laura D'Andrea, Igor V. Komarov, David E. Gloriam, Anders A. Jensen, Christophe Stove (UGent) and Jesper L. Kristensen

(2022) JOURNAL OF MEDICINAL CHEMISTRY. 65(18). p.12031-12043
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The expanding role of chemistry in optimizing proteins for human health applications

Bart Roman (UGent)

(2021) JOURNAL OF MEDICINAL CHEMISTRY. 64(11). p.7179-7188
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2-((3,5-Dinitrobenzyl)thio)quinazolinones : potent antimycobacterial agents activated by deazaflavin (F420)-dependent nitroreductase (Ddn)

Yanlin Jian, He Eun Forbes, Fabian Hulpia (UGent) , Martijn Risseeuw (UGent) , Guy Caljon, Hélène Munier-Lehmann, Helena I. M. Boshoff and Serge Van Calenbergh (UGent)

(2021) JOURNAL OF MEDICINAL CHEMISTRY. 64(1). p.440-457
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Revisiting pyrazolo[3,4-d]pyrimidine nucleosides as anti-trypanosoma cruzi and antileishmanial agents

Jakob Bouton, Ludmila Ferreira de Almeida Fiuza, Camila Cardoso Santos, Maria Angela Mazzarella, Maria de Nazaré Correia Soeiro, Louis Maes, Izet Karalic (UGent) , Guy Caljon and Serge Van Calenbergh (UGent)

(2021) JOURNAL OF MEDICINAL CHEMISTRY. 64(7). p.4206-4238
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Pillar[5]arene-based polycationic glyco[2]rotaxanes designed as Pseudomonas aeruginosa antibiofilm agents

Tharwat Mohy El Dine, Ravikumar Jimmidi, Andrei Diaconu, Maude Fransolet, Carine Michiels, Julien De Winter, Emilie Gillon, Anne Imberty, Tom Coenye (UGent) and Stephane P. Vincent

(2021) JOURNAL OF MEDICINAL CHEMISTRY. 64(19). p.14728-14744
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Systematic investigation of lipophilicity modulation by aliphatic fluorination motifs

Benjamin Jeffries, Zhong Wang, Hannah R. Felstead, Jean-Yves Le Questel, James S. Scott, Elisabetta Chiarparin, Jerome Graton and Bruno Linclau (UGent)

(2020) JOURNAL OF MEDICINAL CHEMISTRY. 63(3). p.1002-1031
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Discovery of pyrrolo[2,3-b]pyridine (1,7-dideazapurine) nucleoside analogues as anti-Trypanosoma cruzi agents

Cai Lin, Fabian Hulpia (UGent) , Cristiane França da Silva, Denise da Gama Jaén Batista, Kristof Van Hecke (UGent) , Louis Maes, Guy Caljon, Maria de Nazaré Correia Soeiro and Serge Van Calenbergh (UGent)

(2019) JOURNAL OF MEDICINAL CHEMISTRY. 62(19). p.8847-8865
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Reducing the lipophilicity of perfluoroalkyl groups by CF2-F/CF2-Me or CF3/CH3 exchange

Benjamin Jeffries, Zhong Wang, Jerome Graton, Simon D. Holland, Thomasin Brind, Ryan D. R. Greenwood, Jean-Yves Le Questel, James S. Scott, Elisabetta Chiarparin and Bruno Linclau (UGent)

(2018) JOURNAL OF MEDICINAL CHEMISTRY. 61(23). p.10602-10618

Academic Bibliography

Dual-acting small molecules : subtype-selective cannabinoid receptor 2 agonist/butyrylcholinesterase inhibitor hybrids show neuroprotection in an Alzheimer's disease mouse model

The zinc-binding group effect : lessons from non-hydroxamic acid vorinostat analogs

Discovery of ss-arrestin-biased 25CN-NBOH-derived 5-HT2A receptor agonists

The expanding role of chemistry in optimizing proteins for human health applications

2-((3,5-Dinitrobenzyl)thio)quinazolinones : potent antimycobacterial agents activated by deazaflavin (F420)-dependent nitroreductase (Ddn)

Revisiting pyrazolo[3,4-d]pyrimidine nucleosides as anti-trypanosoma cruzi and antileishmanial agents

Pillar[5]arene-based polycationic glyco[2]rotaxanes designed as Pseudomonas aeruginosa antibiofilm agents

Systematic investigation of lipophilicity modulation by aliphatic fluorination motifs

Discovery of pyrrolo[2,3-b]pyridine (1,7-dideazapurine) nucleoside analogues as anti-Trypanosoma cruzi agents

Reducing the lipophilicity of perfluoroalkyl groups by CF2-F/CF2-Me or CF3/CH3 exchange

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