Ghent University Academic Bibliography

Journal Article
A1
open access

Synthesis and functional screening of novel inhibitors targeting the HDAC6 zinc finger ubiquitin-binding domain

Silke Geurs, Eleni Staessens (UGent) , Kato Bredael (UGent) , Stefaan Borghgraef, Jordy De Ridder, Leentje Persoons, Steven De Jonghe, Dominique Schols, Mandeep K. Mann, Rachel J. Harding, et al.

(2025) EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. 285.

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Journal Article
A1
open access

Repurposing of monocyclic β-lactams as anti-inflammatory agents : the case of new ferrocene-azetidin-2-one hybrids

Marija S. Gencic, Nikola M. Stojanovic, Jelena M. Denic, Zorica Z. Stojanovic-Radicc, Predrag Stojanovic, Kristof Van Hecke (UGent) , Ljiljana S. Jovanovic, Marija Vukelic Nikolicg, Tatjana Jevtovic-Stoimenovh, Niko S. Radulovic, et al.

(2024) EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. 280.

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Journal Article
A1
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Acyloxymethyl and alkoxycarbonyloxymethyl prodrugs of a fosmidomycin surrogate as antimalarial and antibacterial agents

Charlotte Courtens, Frits van Charante, Thibaut Quennesson (UGent) , Martijn Risseeuw (UGent) , Paul Cos, Guy Caljon, Tom Coenye (UGent) and Serge Van Calenbergh (UGent)

(2023) EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. 245(1).

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Development of teixobactin analogues containing hydrophobic, non-proteogenic amino acids that are highly potent against multidrug-resistant bacteria and biofilms

Anish Parmar, Rajamani Lakshminarayanan, Abhishek Iyer (UGent) , Eunice Tze Leng Goh, Tsz Ying To, Joey Kuok Hoong Yam, Liang Yang, Enas Newire, Maria C. Robertson, Stephen H. Prior, et al.

(2023) EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. 261.

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Journal Article
A1
open access

Targeted AURKA degradation : towards new therapeutic agents for neuroblastoma

Muhammad Rishfi (UGent) , Simon Krols (UGent) , Fien Martens (UGent) , Sarah-Lee Bekaert (UGent) , Ellen Sanders (UGent) , Aline Eggermont (UGent) , Fanny De Vloed (UGent) , Joshua Robert Goulding (UGent) , Martijn Risseeuw (UGent) , Jan Molenaar, et al.

(2023) EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. 247.

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Journal Article
A1
open access

Exploration of 6-methyl-7-(hetero)aryl-7-deazapurine ribonucleosides as antileishmanial agents

Cai Lin, Izet Karalic (UGent) , An Matheeussen, Pim-Bart Feijens, Fabian Hulpia (UGent) , Louis Maes, Guy Caljon and Serge Van Calenbergh (UGent)

(2022) EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. 237.

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A(3) adenosine receptor agonists containing dopamine moieties for enhanced interspecies affinity

Dilip K. Tosh, Veronica Salmaso, Ryan G. Campbell, Harsha Rao, Amelia Bitant, Eline Pottie (UGent) , Christophe Stove (UGent) , Naili Liu, Oksana Gavrilova, Zhan-Guo Gao, et al.

(2022) EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. 228.

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Journal Article
A1
open access

N6-modification of 7-deazapurine nucleoside analogues as anti-Trypanosoma cruzi and anti-Leishmania agents : structure-activity relationship exploration and in vivo evaluation

Cai Lin, Denise da Gama Jaén Batista, Ana Lia Mazzeti, Roberson Donola Girão, Gabriel Melo de Oliveira, Izet Karalic (UGent) , Fabian Hulpia, Maria de Nazaré C. Soeiro, Louis Maes, Guy Caljon, et al.

(2022) EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. 231.

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Journal Article
A1
open access

Synthesis and evaluation of 3′-fluorinated 7-deazapurine nucleosides as antikinetoplastid agents

Jakob Bouton, Arno Furquim d'Almeida, Louis Maes, Guy Caljon, Serge Van Calenbergh (UGent) and Fabian Hulpia (UGent)

(2021) EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. 216.

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Journal Article
A1
open access

Synthesis and evaluation of a collection of purine-like C-nucleosides as antikinetoplastid agents

Jakob Bouton, Louis Maes, Izet Karalic (UGent) , Guy Caljon and Serge Van Calenbergh (UGent)

(2021) EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. 212.

Academic Bibliography

Synthesis and functional screening of novel inhibitors targeting the HDAC6 zinc finger ubiquitin-binding domain

Repurposing of monocyclic β-lactams as anti-inflammatory agents : the case of new ferrocene-azetidin-2-one hybrids

Acyloxymethyl and alkoxycarbonyloxymethyl prodrugs of a fosmidomycin surrogate as antimalarial and antibacterial agents

Development of teixobactin analogues containing hydrophobic, non-proteogenic amino acids that are highly potent against multidrug-resistant bacteria and biofilms

Targeted AURKA degradation : towards new therapeutic agents for neuroblastoma

Exploration of 6-methyl-7-(hetero)aryl-7-deazapurine ribonucleosides as antileishmanial agents

A(3) adenosine receptor agonists containing dopamine moieties for enhanced interspecies affinity

N6-modification of 7-deazapurine nucleoside analogues as anti-Trypanosoma cruzi and anti-Leishmania agents : structure-activity relationship exploration and in vivo evaluation

Synthesis and evaluation of 3′-fluorinated 7-deazapurine nucleosides as antikinetoplastid agents

Synthesis and evaluation of a collection of purine-like C-nucleosides as antikinetoplastid agents

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