Ghent University Academic Bibliography

Journal Article

Acyloxymethyl and alkoxycarbonyloxymethyl prodrugs of a fosmidomycin surrogate as antimalarial and antibacterial agents

Charlotte Courtens, Frits van Charante (UGent) , Thibaut Quennesson, Martijn Risseeuw (UGent) , Paul Cos, Guy Caljon, Tom Coenye (UGent) and Serge Van Calenbergh (UGent)

(2023) EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. 245.

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Journal Article
A1
open access

Targeted AURKA degradation : towards new therapeutic agents for neuroblastoma

Muhammad Rishfi (UGent) , Simon Krols (UGent) , Fien Martens (UGent) , Sarah-Lee Bekaert (UGent) , Ellen Sanders (UGent) , Aline Eggermont (UGent) , Fanny De Vloed (UGent) , Joshua Robert Goulding (UGent) , Martijn Risseeuw (UGent) , Jan Molenaar, et al.

(2023) EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. 247.

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Journal Article
A1
open access

Exploration of 6-methyl-7-(hetero)aryl-7-deazapurine ribonucleosides as antileishmanial agents

Cai Lin (UGent) , Izet Karalic (UGent) , An Matheeussen, Pim-Bart Feijens, Fabian Hulpia (UGent) , Louis Maes, Guy Caljon and Serge Van Calenbergh (UGent)

(2022) EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. 237.

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A(3) adenosine receptor agonists containing dopamine moieties for enhanced interspecies affinity

Dilip K. Tosh, Veronica Salmaso, Ryan G. Campbell, Harsha Rao, Amelia Bitant, Eline Pottie (UGent) , Christophe Stove (UGent) , Naili Liu, Oksana Gavrilova, Zhan-Guo Gao, et al.

(2022) EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. 228.

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Journal Article
A1
open access

N6-modification of 7-deazapurine nucleoside analogues as anti-Trypanosoma cruzi and anti-Leishmania agents : structure-activity relationship exploration and in vivo evaluation

Cai Lin (UGent) , Denise da Gama Jaén Batista, Ana Lia Mazzeti, Roberson Donola Girão, Gabriel Melo de Oliveira, Izet Karalic (UGent) , Fabian Hulpia, Maria de Nazaré C. Soeiro, Louis Maes, Guy Caljon, et al.

(2022) EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. 231.

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Journal Article
A1
open access

Recent contributions of quinolines to antimalarial and anticancer drug discovery research

Tim Van de Walle, Lore Cools, Sven Mangelinckx (UGent) and Matthias D'hooghe (UGent)

(2021) EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. 226.

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Journal Article
A1
open access

Synthesis and evaluation of 3′-fluorinated 7-deazapurine nucleosides as antikinetoplastid agents

Jakob Bouton, Arno Furquim d'Almeida, Louis Maes, Guy Caljon, Serge Van Calenbergh (UGent) and Fabian Hulpia (UGent)

(2021) EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. 216.

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Journal Article
A1
open access

Synthesis and evaluation of a collection of purine-like C-nucleosides as antikinetoplastid agents

Jakob Bouton, Louis Maes, Izet Karalic (UGent) , Guy Caljon and Serge Van Calenbergh (UGent)

(2021) EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. 212.

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Discovery of a true bivalent dopamine D2 receptor agonist

Mingcheng Qian, Adrián Ricarte, Elise Wouters, James A.R. Dalton, Martijn Risseeuw (UGent) , Jesús Giraldo and Serge Van Calenbergh (UGent)

(2021) EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. 212.

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Structure-aided optimization of non-nucleoside M. tuberculosis thymidylate kinase inhibitors

Lijun Song (UGent) , Romain Merceron (UGent) , Fabian Hulpia (UGent) , Ainhoa Lucia, Begona Gracia, Yanlin Jian, Martijn Risseeuw (UGent) , Toon Verstraelen (UGent) , Paul Cos, Jose A. Ainsa, et al.

(2021) EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. 225.

Academic Bibliography

Acyloxymethyl and alkoxycarbonyloxymethyl prodrugs of a fosmidomycin surrogate as antimalarial and antibacterial agents

Targeted AURKA degradation : towards new therapeutic agents for neuroblastoma

Exploration of 6-methyl-7-(hetero)aryl-7-deazapurine ribonucleosides as antileishmanial agents

A(3) adenosine receptor agonists containing dopamine moieties for enhanced interspecies affinity

N6-modification of 7-deazapurine nucleoside analogues as anti-Trypanosoma cruzi and anti-Leishmania agents : structure-activity relationship exploration and in vivo evaluation

Recent contributions of quinolines to antimalarial and anticancer drug discovery research

Synthesis and evaluation of 3′-fluorinated 7-deazapurine nucleosides as antikinetoplastid agents

Synthesis and evaluation of a collection of purine-like C-nucleosides as antikinetoplastid agents

Discovery of a true bivalent dopamine D2 receptor agonist

Structure-aided optimization of non-nucleoside M. tuberculosis thymidylate kinase inhibitors

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