Academic Bibliography

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Structure-activity relationship in monosaccharide-based Toll-like receptor 4 (TLR4) antagonists

Fabio A Facchini, Lenny Zaffaroni, Alberto Minotti, Silvia Rapisarda, Valentina Calabrese, Matilde Forcella, Paola Fusi, Cristina Airoldi, Carlotta Ciaramelli, Jean-Marc Billod, et al.

(2018) JOURNAL OF MEDICINAL CHEMISTRY. 61(7). p.2895-2909
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Structure Guided Lead Generation toward Nonchiral M. tuberculosis Thymidylate Kinase Inhibitors

Lijun Song, Romain Merceron, Begoña Gracia, Ainhoa Lucía Quintana, Martijn D. P. Risseeuw, Fabian Hulpia, Paul Cos, José A. Aínsa, Hélène Munier-Lehmann, Savvas N. Savvides, et al.

(2018) J. Med. Chem.. 61(7).
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Medicinal chemistry and use of myosin II inhibitor (S)-blebbistatin and its derivatives

Bart Roman (UGent), Sigrid Verhasselt (UGent) and Christian Stevens (UGent)

(2018) JOURNAL OF MEDICINAL CHEMISTRY.
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Tozasertib analogues as inhibitors of necroptotic cell death

Sam Hofmans, Lars Devisscher, Sofie Martens (UGent), Dries Van Rompaey, Kenneth Goossens, Tatyana Divert (UGent), Wim Nerinckx (UGent), Nozomi Takahashi (UGent), Hans De Winter, Pieter Van der Veken, et al.

(2018) JOURNAL OF MEDICINAL CHEMISTRY. 61(5). p.1895-1920
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Design and syntheses of highly potent teixobactin analogues against Staphylococcus aureus, methicillin-resistant Staphylococcus aureus (MRSA), vancomycin-resistant Enterococci (VRE) in vitro and in vivo

Anish Parmar, Rajamani Lakshminarayanan, Abhishek Iyer (UGent), Venkatesh Mayandi, Eunice Tze Leng Goh, Daniel G Lloyd, Madhavi Latha S Chalasani, Navin Kumar Verma, Stephen H Prior, Roger W Beuerman, et al.

(2018) JOURNAL OF MEDICINAL CHEMISTRY. 61(5). p.2009-2017
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Determination of in vitro and in silico indexes for the modeling of blood-brain barrier partitioning of drugs via micellar and immobilized artificial membrane liquid chromatography

Giacomo Russo (UGent), Lucia Grumetto, Roman Szucs (UGent), Francesco Barbato and Frederic Lynen (UGent)

(2017) JOURNAL OF MEDICINAL CHEMISTRY. 60(9). p.3739-3754
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Discovery of mycobacterium tuberculosis InhA inhibitors by binding sites comparison and ligands prediction

Tanja Štular, Samo Lešnik, Kaja Rožman, Julia Schink, Mitja Zdouc, An Ghysels (UGent), Feng Liu, Courtney C Aldrich, V Joachim Haupt, Sebastian Salentin, et al.

(2016) JOURNAL OF MEDICINAL CHEMISTRY . 59(24). p.11069-11078
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Novel ferroptosis inhibitors with improved potency and ADME properties

Sam Hofmans, Tom Vanden Berghe (UGent), Lars Devisscher, Behrouz Hassannia (UGent), Sophie Lyssens, Jurgen Joossens, Pieter Van Der Veken, Peter Vandenabeele (UGent) and Koen Augustyns

(2016) JOURNAL OF MEDICINAL CHEMISTRY. 59(5). p.2041-2053
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Synthesis and bioactivity of β-substituted fosmidomycin analogues targeting 1-deoxy-D-xylulose-5-phosphate reductoisomerase

René Chofor, Sanjeewani Sooriyaarachchi, Martijn Risseeuw (UGent), Terese Bergfors, Jenny Pouyez, Chinchu Johny, Amanda Haymond, Annelien Everaert, Cynthia S Dowd, Louis Maes, et al.

(2015) JOURNAL OF MEDICINAL CHEMISTRY. 58(7). p.2988-3001
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Structural investigation of B-Raf paradox breaker and inducer inhibitors

Rohit Arora, Michela Di Michele, Elisabeth Stes, Elien Vandermarliere (UGent), Lennart Martens (UGent), Kris Gevaert (UGent), Erika Van Heerde, Joannes TM Linders, Dirk Brehmer, Edgar Jacoby, et al.

(2015) JOURNAL OF MEDICINAL CHEMISTRY. 58(4). p.1818-1831

Academic Bibliography

Biblio has been updated

Structure-activity relationship in monosaccharide-based Toll-like receptor 4 (TLR4) antagonists

Structure Guided Lead Generation toward Nonchiral M. tuberculosis Thymidylate Kinase Inhibitors

Medicinal chemistry and use of myosin II inhibitor (S)-blebbistatin and its derivatives

Tozasertib analogues as inhibitors of necroptotic cell death

Design and syntheses of highly potent teixobactin analogues against Staphylococcus aureus, methicillin-resistant Staphylococcus aureus (MRSA), vancomycin-resistant Enterococci (VRE) in vitro and in vivo

Determination of in vitro and in silico indexes for the modeling of blood-brain barrier partitioning of drugs via micellar and immobilized artificial membrane liquid chromatography

Discovery of mycobacterium tuberculosis InhA inhibitors by binding sites comparison and ligands prediction

Novel ferroptosis inhibitors with improved potency and ADME properties

Synthesis and bioactivity of β-substituted fosmidomycin analogues targeting 1-deoxy-D-xylulose-5-phosphate reductoisomerase

Structural investigation of B-Raf paradox breaker and inducer inhibitors

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