Ghent University Academic Bibliography

Journal Article
A1
open access

Report on a new opioid NPS : chemical and in vitro functional characterization of a structural isomer of the MT-45 derivative diphenpipenol

Annelies Cannaert (UGent) , Fabian Hulpia (UGent) , Martijn Risseeuw (UGent) , Katleen Van Uytfanghe (UGent) , Eric Deconinck, Serge Van Calenbergh (UGent) , Peter Blanckaert and Christophe Stove (UGent)

(2021) JOURNAL OF ANALYTICAL TOXICOLOGY. 45(2). p.134-140

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2-((3,5-Dinitrobenzyl)thio)quinazolinones : potent antimycobacterial agents activated by deazaflavin (F420)-dependent nitroreductase (Ddn)

Yanlin Jian (UGent) , He Eun Forbes, Fabian Hulpia (UGent) , Martijn Risseeuw (UGent) , Guy Caljon, Hélène Munier-Lehmann, Helena I. M. Boshoff and Serge Van Calenbergh (UGent)

(2021) JOURNAL OF MEDICINAL CHEMISTRY. 64(1). p.440-457

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Journal Article
A1
open access

RUNX2 regulates leukemic cell metabolism and chemotaxis in high-risk T cell acute lymphoblastic leukemia

Filip Matthijssens (UGent) , Nitesh D. Sharma, Monique Nysus, Christian K. Nickl, Huining Kang, Dominique R. Perez, Béatrice Lintermans (UGent) , Wouter Van Loocke (UGent) , Juliette Roels (UGent) , Sofie Peirs (UGent) , et al.

(2021) JOURNAL OF CLINICAL INVESTIGATION. 131(6).

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Structure-aided optimization of non-nucleoside M. tuberculosis thymidylate kinase inhibitors

Lijun Song (UGent) , Romain Merceron (UGent) , Fabian Hulpia (UGent) , Ainhoa Lucia, Begona Gracia, Yanlin Jian (UGent) , Martijn Risseeuw (UGent) , Toon Verstraelen (UGent) , Paul Cos, Jose A. Ainsa, et al.

(2021) EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. 225.

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Discovery of a true bivalent dopamine D2 receptor agonist

Mingcheng Qian, Adrián Ricarte, Elise Wouters, James A.R. Dalton, Martijn Risseeuw (UGent) , Jesús Giraldo and Serge Van Calenbergh (UGent)

(2021) EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. 212.

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Synthesis and structure activity relationships of cyanopyridone based anti-tuberculosis agents

Yanlin Jian (UGent) , Fabian Hulpia (UGent) , Martijn Risseeuw (UGent) , He Eun Forbes, Hélène Munier-Lehmann, Guy Caljon, Helena I. M. Boshoff and Serge Van Calenbergh (UGent)

(2020) EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. 201.

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Journal Article
A1
open access

1-(1-Arylethylpiperidin-4-yl)thymine analogs as antimycobacterial TMPK inhibitors

Yanlin Jian (UGent) , Fabian Hulpia (UGent) , Martijn Risseeuw (UGent) , He Eun Forbes, Guy Caljon, Hélène Munier-Lehmann, Helena I. M. Boshoff and Serge Van Calenbergh (UGent)

(2020) MOLECULES. 25(12).

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Synthetic rhamnose glycopolymer cell-surface receptor for endogenous antibody recruitment

Ruben De Coen (UGent) , Lutz Nuhn, Chamani Perera, Maria Arista-Romero, Martijn Risseeuw (UGent) , Alec Freyn, Raffael Nachbagauer, Lorenzo Albertazzi, Serge Van Calenbergh (UGent) , David A. Spiegel, et al.

(2020) BIOMACROMOLECULES. 21(2). p.793-802

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Journal Article
A1
open access

Design, synthesis and characterization of a new series of fluorescent metabotropic glutamate receptor type 5 negative allosteric modulators

Víctor Fernández-Dueñas, Mingcheng Qian, Josep Argerich, Carolina Amaral, Martijn Risseeuw (UGent) , Serge Van Calenbergh (UGent) and Francisco Ciruela

(2020) MOLECULES. 25(7).

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Journal Article
A1
open access

Endeavors towards transformation of M. tuberculosis thymidylate kinase (MtbTMPK) inhibitors into potential antimycobacterial agents

Yanlin Jian (UGent) , Romain Merceron (UGent) , Steven De Munck (UGent) , He Eun Forbes, Fabian Hulpia (UGent) , Martijn Risseeuw (UGent) , Kristof Van Hecke (UGent) , Savvas Savvides (UGent) , Hélène Munier-Lehmann, Helena I. M. Boshoff, et al.

(2020) EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. 206.

Academic Bibliography

Report on a new opioid NPS : chemical and in vitro functional characterization of a structural isomer of the MT-45 derivative diphenpipenol

2-((3,5-Dinitrobenzyl)thio)quinazolinones : potent antimycobacterial agents activated by deazaflavin (F420)-dependent nitroreductase (Ddn)

RUNX2 regulates leukemic cell metabolism and chemotaxis in high-risk T cell acute lymphoblastic leukemia

Structure-aided optimization of non-nucleoside M. tuberculosis thymidylate kinase inhibitors

Discovery of a true bivalent dopamine D2 receptor agonist

Synthesis and structure activity relationships of cyanopyridone based anti-tuberculosis agents

1-(1-Arylethylpiperidin-4-yl)thymine analogs as antimycobacterial TMPK inhibitors

Synthetic rhamnose glycopolymer cell-surface receptor for endogenous antibody recruitment

Design, synthesis and characterization of a new series of fluorescent metabotropic glutamate receptor type 5 negative allosteric modulators

Endeavors towards transformation of M. tuberculosis thymidylate kinase (MtbTMPK) inhibitors into potential antimycobacterial agents

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