Ghent University Academic Bibliography

Journal Article
A1
open access

Report on a new opioid NPS : chemical and in vitro functional characterization of a structural isomer of the MT-45 derivative diphenpipenol

Annelies Cannaert (UGent) , Fabian Hulpia (UGent) , Martijn Risseeuw (UGent) , Katleen Van Uytfanghe (UGent) , Eric Deconinck, Serge Van Calenbergh (UGent) , Peter Blanckaert and Christophe Stove (UGent)

(2021) JOURNAL OF ANALYTICAL TOXICOLOGY. 45(2). p.134-140

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Journal Article
A1
open access

RUNX2 regulates leukemic cell metabolism and chemotaxis in high-risk T cell acute lymphoblastic leukemia

Filip Matthijssens (UGent) , Nitesh D. Sharma, Monique Nysus, Christian K. Nickl, Huining Kang, Dominique R. Perez, Béatrice Lintermans (UGent) , Wouter Van Loocke (UGent) , Juliette Roels (UGent) , Sofie Peirs (UGent) , et al.

(2021) JOURNAL OF CLINICAL INVESTIGATION. 131(6).

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2-((3,5-Dinitrobenzyl)thio)quinazolinones : potent antimycobacterial agents activated by deazaflavin (F420)-dependent nitroreductase (Ddn)

Yanlin Jian (UGent) , He Eun Forbes, Fabian Hulpia (UGent) , Martijn Risseeuw (UGent) , Guy Caljon, Hélène Munier-Lehmann, Helena I. M. Boshoff and Serge Van Calenbergh (UGent)

(2021) JOURNAL OF MEDICINAL CHEMISTRY. 64(1). p.440-457

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6‐methyl‐7‐aryl‐7‐deazapurine nucleosides as anti‐trypanosoma cruzi agents : structure‐activity relationship and in vivo efficacy

Cai Lin (UGent) , Ludmila Ferreira de Almeida Fiuza, Camila Cardoso Santos, Daniela Ferreira Nunes, Otacílio Cruz Moreira, Jakob Bouton (UGent) , Izet Karalic (UGent) , Louis Maes, Guy Caljon, Fabian Hulpia (UGent) , et al.

(2021) CHEMMEDCHEM. 16(14). p.2231-2253

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Synthesis and evaluation of 3′-fluorinated 7-deazapurine nucleosides as antikinetoplastid agents

Jakob Bouton (UGent) , Arno Furquim d'Almeida, Louis Maes, Guy Caljon, Serge Van Calenbergh (UGent) and Fabian Hulpia (UGent)

(2021) EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. 216.

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Revisiting pyrazolo[3,4-d]pyrimidine nucleosides as anti-trypanosoma cruzi and antileishmanial agents

Jakob Bouton (UGent) , Ludmila Ferreira de Almeida Fiuza, Camila Cardoso Santos, Maria Angela Mazzarella, Maria de Nazaré Correia Soeiro, Louis Maes, Izet Karalic (UGent) , Guy Caljon and Serge Van Calenbergh (UGent)

(2021) JOURNAL OF MEDICINAL CHEMISTRY. 64(7). p.4206-4238

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Journal Article
A1
open access

4E interacting protein as a potential novel drug target for nucleoside analogues in Trypanosoma brucei

Dorien Mabille, Camila Cardoso Santos, Rik Hendrickx, Mathieu Claes, Peter Takac, Christine Clayton, Sarah Hendrickx, Fabian Hulpia (UGent) , Louis Maes, Serge Van Calenbergh (UGent) , et al.

(2021) MICROORGANISMS. 9(4).

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Synthesis and evaluation of a collection of purine-like C-nucleosides as antikinetoplastid agents

Jakob Bouton (UGent) , Louis Maes, Izet Karalic (UGent) , Guy Caljon and Serge Van Calenbergh (UGent)

(2021) EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. 212.

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Discovery of a true bivalent dopamine D2 receptor agonist

Mingcheng Qian, Adrián Ricarte, Elise Wouters, James A.R. Dalton, Martijn Risseeuw (UGent) , Jesús Giraldo and Serge Van Calenbergh (UGent)

(2021) EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. 212.

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Sustainability in drug discovery

Evelien Wynendaele (UGent) , Christophe Furman, Bartosz Wielgomas, Per Larsson, Eelko Hak, Thomas Block (UGent) , Serge Van Calenbergh (UGent) , Nicolas Willand, Michal Markuszewski, Luke R. Odell, et al.

(2021) MEDICINE IN DRUG DISCOVERY. 12.

Academic Bibliography

Report on a new opioid NPS : chemical and in vitro functional characterization of a structural isomer of the MT-45 derivative diphenpipenol

RUNX2 regulates leukemic cell metabolism and chemotaxis in high-risk T cell acute lymphoblastic leukemia

2-((3,5-Dinitrobenzyl)thio)quinazolinones : potent antimycobacterial agents activated by deazaflavin (F420)-dependent nitroreductase (Ddn)

6‐methyl‐7‐aryl‐7‐deazapurine nucleosides as anti‐trypanosoma cruzi agents : structure‐activity relationship and in vivo efficacy

Synthesis and evaluation of 3′-fluorinated 7-deazapurine nucleosides as antikinetoplastid agents

Revisiting pyrazolo[3,4-d]pyrimidine nucleosides as anti-trypanosoma cruzi and antileishmanial agents

4E interacting protein as a potential novel drug target for nucleoside analogues in Trypanosoma brucei

Synthesis and evaluation of a collection of purine-like C-nucleosides as antikinetoplastid agents

Discovery of a true bivalent dopamine D2 receptor agonist

Sustainability in drug discovery

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