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Photo-induced crosslinking uncovers an antiparallel strand orientation in heterodimeric (EIAALEK)(3)/(KIAALKE)(3) and (EIAALEK)(3)/(RIAALRE)(3) coiled-coil systems
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- Journal Article
- open access
Dithioallyl cation (3+2) cycloadditions under aprotic reaction conditions: rapid access to spiro-fused cyclopentane scaffolds
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GlyConnect-Ugi : site-selective, multi-component glycoprotein conjugations through GlycoDelete expressed glycans
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Nucleotides bearing aminophenyl- or aminonaphthyl-3-methoxychromone solvatochromic fluorophores for the enzymatic construction of DNA probes for the detection of protein–DNA binding
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Enzymatic glycosylation involving fluorinated carbohydrates
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Caspase-3 probes for PET imaging of apoptotic tumor response to anticancer therapy
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Gold(I) catalysed regio- and stereoselective intermolecular hydroamination of internal alkynes : towards functionalised azoles
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Synthesis of vicinal dideoxy-difluorinated galactoses
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Theoretical insight into the regioselective ring-expansions of bicyclic aziridinium ions
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Domino reaction of a gold catalyzed 5-endo-dig cyclization and a [3,3]-sigmatropic rearrangement towards polysubstituted pyrazoles
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Cobalt carbonyl-catalyzed carbonylation of functionalized aziridines to versatile β-lactam building blocks
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Synthesis of C6′′-modified α-C-GalCer analogues as mouse and human iNKT cell agonists
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Singlet oxygen-mediated one-pot chemoselective peptide-peptide ligation
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Decoration of trastuzumab with short oligonucleotides : synthesis and detailed characterization
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Porphyrin-based photosensitizers and their DNA conjugates for singlet oxygen induced nucleic acid interstrand crosslinking
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Carboxylate isosteres for caspase inhibitors : the acylsulfonamide case revisited
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- Journal Article
- A1
- open access
Discovery of (S)-3′-hydroxyblebbistatin and (S)-3′-aminoblebbistatin : polar myosin II inhibitors with superior research tool properties
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Direct subphthalocyanine conjugation to bombesin vs. indirect conjugation to its lipidic nanocarrier
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Triflate-functionalized calix[6]arenes as versatile building-blocks : application to the synthesis of an inherently chiral Zn(II) complex
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Evaluation of the transfection efficacies of quaternary ammonium salts prepared from sophorolipids
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Bioconjugation: using selective chemistry to enhance the properties of proteins and peptides as therapeutics and carriers
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- Journal Article
- A1
- open access
Diastereoselective synthesis of 3-acetoxy-4-(3-aryloxiran-2-yl)azetidin-2-ones and their transformation into 3,4-oxolane-fused bicyclic β-lactams
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- Journal Article
- A1
- open access
Synthesis and SAR assessment of novel Tubathian analogs in the pursuit of potent and selective HDAC6 inhibitors
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Design, synthesis and biological activities of new brassinosteroid analogues with a phenyl group in the side chain
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The development of a short route to the API ropinirole hydrochloride
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Phosphonamide pyrabactin analogues as abscisic acid agonists
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Tuning temperature responsive poly(2-alkyl-2-oxazoline)s by supramolecular host-guest interactions
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Synthesis of 2-aryl-3-(2-cyanoethyl)aziridines and their chemical and enzymatic hydrolysis towards γ-lactams and γ-lactones
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Antibodies armed with photosensitizers: from chemical synthesis to photobiological applications
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Cyclodextrin-peptide conjugates for sequence specific DNA binding
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Oxidative α,ω-diyne coupling as an approach towards novel peptidic macrocycles
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Evaluation of the antibacterial and antibiofilm activities of novel CRAMP-vancomycin conjugates with diverse linkers
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Stapling monomeric GCN4 peptides allows for DNA binding and enhanced cellular uptake
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Asymmetric synthesis of chloroisothreonine derivatives via syn-stereoselective Mannich-type additions across N-sulfinyl-α-chloroimines
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[Pd(mu-Cl)Cl(IPr*)](2) : a highly hindered pre-catalyst for the synthesis of tetra-ortho-substituted biaryls via Grignard reagent cross-coupling
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Water-soluble NHC-Cu catalysts : applications in click chemistry, bioconjugation and mechanistic analysis
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Porphyrin conjugated with serum albumins and monoclonal antibodies boosts efficiency in targeted destruction of human bladder cancer cells
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A mildly inducible and selective cross-link methodology for RNA duplexes
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Regioselective ruthenium catalysed H-D exchange using D2O as the deuterium source
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Iridium(I) hydroxides in catalysis : rearrangement of allylic alcohols to ketones
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Synthesis and structure of large difluoromethylene containing alicycles by ring closing metathesis (RCM)
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- Journal Article
- A1
- open access
Radical-mediated nitrile translocation as the key step in the stereoselective transformation of 2-(4-chloro-2-cyanobutyl)aziridines to methyl cis-(1-arylmethyl-4-phenylpiperidin-2-yl)acetates
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Aromatic capping surprisingly stabilizes furan moieties in peptides against acidic degradation
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Homoselenacalix[4]arenes : synthetic exploration and metallosupramolecular chemistry
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A convenient synthesis of difficult medium-sized cyclic peptides by Staudinger mediated ring-closure
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Asymmetric synthesis of α,β-diamino acid derivatives with an aziridine-, azetidine- and γ-lactone-skeleton via Mannich-type additions across α-chloro-N-sulfinylimines
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Fast RNA conjugations on solid phase by strain-promoted cycloadditions
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Chiral imidate-ferrocenylphosphanes: synthesis and application as P,N-ligands in iridium(I)-catalyzed hydrogenation of unfunctionalized and poorly functionalized olefins
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- Journal Article
- A1
- open access
Synthesis of novel β-aminocyclobutanecarboxylic acid derivatives by a solvent-free aza-Michael addition and subsequent ring closure
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Synthesis, modeling and evaluation of 3'-(1-aryl-1H-tetrazol-5-ylamino)-substituted 3'-deoxythymidine derivatives as potent and selective human mitochondrial thymidine kinase inhibitors
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A combined mechanistic and computational study of the gold(I)-catalyzed formation of substituted indenes
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Well-defined [Rh(NHC)(OH)] complexes enabling the conjugate addition of arylboronic acids to α,β-unsaturated ketones
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- Journal Article
- A1
- open access
New general synthesis of alpha-alkoxyketones via alpha'-alkylation, alpha-alkylation and alpha,alpha'-dialkylation of alpha-alkoxyketimines
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Synthesis of 1-substituted 1,2,3,4-tetrahydrobenz[g]isoquinoline-5,10-diones
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Gold(III) chloride catalysed synthesis of 5-alkylidene-dihydrothiazoles
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Divergent synthetic approach to 6''-modified α-GalCer analogues
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- Journal Article
- A1
- open access
Straightforward synthesis of 1-alkyl-2-(trifluoromethyl)aziridines starting from 1,1,1-trifluoroacetone
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- Journal Article
- A1
- open access
Stereoselective synthesis of trans- and cis-2-aryl-3-(hydroxymethyl)aziridines through transformation of 4-aryl-3-chloro-β-lactams and study of their ring opening
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Asymmetric synthesis of new chiral N-sulfinyl 2,2-disubstituted aziridines by Grignard additions across alpha-chloro N-sulfinyl ketimines
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Synthesis of C-6-substituted uridine phosphonates through aerobic ligand-free Suzuki-Miyaura cross-coupling
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Synthesis of 5-amino- and 5-hydroxy-3,3-difluoropiperidines
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Experimental and computational study of the ring opening of tricyclic oxanorbornenes to polyhydro isoindole phosphonates
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Synthesis of aminomethylated 4-fluoropiperidines and 3-fluoropyrrolidines
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- Journal Article
- A1
- open access
Microwave-assisted regioselective ring opening of non-activated aziridines by lithium aluminium hydride
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Towards the conformational mimicry of the measles virus HNE loop: design, synthesis and biological evaluation of a cyclic bile acid-peptide conjugate
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A new entry into cis-3-amino-2-methylpyrrolidines via ring expansion of 2-(2-hydroxyethyl)-3-methylaziridines
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A new approach towards 1-phenyl and 1-benzyl substituted 2-(aminomethyl)cyclopropanecarboxamides as novel derivatives of the antidepressant Milnacipran
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Enantioselective synthesis of tetrafluorinated ribose and fructose
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Nonenzymic polycyclisation of analogues of oxidosqualene with a preformed C-ring
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Reactivity of N-(omega-haloalkyl)-beta-lactams with regard to lithium aluminium hydride: novel synthesis of 1-(1-aryl-3-hydroxypropyl)aziridines and 3-aryl-3-(N-propylamino)propan-1-ols
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Electrophile-induced bromocyclization of gamma,delta-unsaturated ketimines to intermediate I-pyrrolinium salts and their selective conversion into novel 5-alkoxymethyl-2-aryl-3-chloropyrroles and 2-aroylpyrroles
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Regio- and stereocontrolled synthesis of novel 3-sulfonamido-2,3,4,5-tetrahydro-1,5-benzothiazepines from 2-(bromomethyl)- or 2-(sulfonyloxymethyl)aziridines
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Glycosynthase activity of hybrid aspen xyloglucan endo-transglycosylase PttXET16-34 nucleophile mutants
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Oxidative reactions of 6-pentyl indolo[3,2-b]carbazole: formation of novel C-C and C-N coupled dimers
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Preparation and relevance of a cross-coupling product between sinapyl alcohol and sinapyl p-hydroxybenzoate
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Synthesis, biological activity, and conformational analysis of CD-ring modified trans-decalin 1 alpha,25-dihydroxyvitamin D analogs
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Synthesis of unprotected and borane-protected cyclic phosphines using Ru- and Mo-based olefin metathesis catalysts
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Ab initio study of the binding of Trichostatin A (TSA) in the active site of Histone Deacetylase Like Protein (HDLP)