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Three-component reaction of a 2-aminoazine, a 2-oxoaldehyde, and a cyclic 1,3-dicarbonyl compound for the synthesis of imidazo[1,2-a]azine derivatives

(2014) ACS COMBINATORIAL SCIENCE. 16(10). p.535-542
Author
Organization
Abstract
A three-component reaction of a 2-aminoazine, a 2-oxoaldehyde, and a cyclic 1,3-dicarbonyl compound providing access toward a novel class of imidazo[1,2-a]azine derivatives was developed and studied. The scope of the process was thoroughly explored under three different reaction conditions resulting in the generation of a small library of title compounds and highlighting the possibility of case-specific approach.
Keywords
ZOLPIDEM, ALPIDEM, 4-TRIAZOLE, 2-AMINOIMIDAZOLES, multicomponent reactions, 2-aminoazines, 2-oxoaldehydes, 1, 3-dicarbonyl compounds, imidazo[1, 2-a]azines, ONE-POT SYNTHESIS, REGIOSELECTIVE SYNTHESIS, MULTICOMPONENT REACTION, EFFICIENT SYNTHESIS, ARYLGLYOXALS, HETEROCYCLES, 2, 3-AMINO-1

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Citation

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MLA
Peshkov, Vsevolod A., et al. “Three-Component Reaction of a 2-Aminoazine, a 2-Oxoaldehyde, and a Cyclic 1,3-Dicarbonyl Compound for the Synthesis of Imidazo[1,2-a]Azine Derivatives.” ACS COMBINATORIAL SCIENCE, vol. 16, no. 10, 2014, pp. 535–42.
APA
Peshkov, V. A., Peshkov, A. A., Pereshivko, O. P., Van Hecke, K., Zamigaylo, L. L., Van der Eycken, E. V., & Gorobets, N. Y. (2014). Three-component reaction of a 2-aminoazine, a 2-oxoaldehyde, and a cyclic 1,3-dicarbonyl compound for the synthesis of imidazo[1,2-a]azine derivatives. ACS COMBINATORIAL SCIENCE, 16(10), 535–542.
Chicago author-date
Peshkov, Vsevolod A, Anatoly A Peshkov, Olga P Pereshivko, Kristof Van Hecke, Lali L Zamigaylo, Erik V Van der Eycken, and Nikolay Yu Gorobets. 2014. “Three-Component Reaction of a 2-Aminoazine, a 2-Oxoaldehyde, and a Cyclic 1,3-Dicarbonyl Compound for the Synthesis of Imidazo[1,2-a]Azine Derivatives.” ACS COMBINATORIAL SCIENCE 16 (10): 535–42.
Chicago author-date (all authors)
Peshkov, Vsevolod A, Anatoly A Peshkov, Olga P Pereshivko, Kristof Van Hecke, Lali L Zamigaylo, Erik V Van der Eycken, and Nikolay Yu Gorobets. 2014. “Three-Component Reaction of a 2-Aminoazine, a 2-Oxoaldehyde, and a Cyclic 1,3-Dicarbonyl Compound for the Synthesis of Imidazo[1,2-a]Azine Derivatives.” ACS COMBINATORIAL SCIENCE 16 (10): 535–542.
Vancouver
1.
Peshkov VA, Peshkov AA, Pereshivko OP, Van Hecke K, Zamigaylo LL, Van der Eycken EV, et al. Three-component reaction of a 2-aminoazine, a 2-oxoaldehyde, and a cyclic 1,3-dicarbonyl compound for the synthesis of imidazo[1,2-a]azine derivatives. ACS COMBINATORIAL SCIENCE. 2014;16(10):535–42.
IEEE
[1]
V. A. Peshkov et al., “Three-component reaction of a 2-aminoazine, a 2-oxoaldehyde, and a cyclic 1,3-dicarbonyl compound for the synthesis of imidazo[1,2-a]azine derivatives,” ACS COMBINATORIAL SCIENCE, vol. 16, no. 10, pp. 535–542, 2014.
@article{5770646,
  abstract     = {A three-component reaction of a 2-aminoazine, a 2-oxoaldehyde, and a cyclic 1,3-dicarbonyl compound providing access toward a novel class of imidazo[1,2-a]azine derivatives was developed and studied. The scope of the process was thoroughly explored under three different reaction conditions resulting in the generation of a small library of title compounds and highlighting the possibility of case-specific approach.},
  author       = {Peshkov, Vsevolod A and Peshkov, Anatoly A and Pereshivko, Olga P and Van Hecke, Kristof and Zamigaylo, Lali L and Van der Eycken, Erik V and Gorobets, Nikolay Yu},
  issn         = {2156-8952},
  journal      = {ACS COMBINATORIAL SCIENCE},
  keywords     = {ZOLPIDEM,ALPIDEM,4-TRIAZOLE,2-AMINOIMIDAZOLES,multicomponent reactions,2-aminoazines,2-oxoaldehydes,1,3-dicarbonyl compounds,imidazo[1,2-a]azines,ONE-POT SYNTHESIS,REGIOSELECTIVE SYNTHESIS,MULTICOMPONENT REACTION,EFFICIENT SYNTHESIS,ARYLGLYOXALS,HETEROCYCLES,2,3-AMINO-1},
  language     = {eng},
  number       = {10},
  pages        = {535--542},
  title        = {Three-component reaction of a 2-aminoazine, a 2-oxoaldehyde, and a cyclic 1,3-dicarbonyl compound for the synthesis of imidazo[1,2-a]azine derivatives},
  url          = {http://dx.doi.org/10.1021/c05000695},
  volume       = {16},
  year         = {2014},
}

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