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Synthesis and biological evaluation of apionucleosides and their protides

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Abstract
We report the synthesis of the A and T 2',3'-dideoxyapionucleosides and their corresponding Pro-Tide derivatives from 1,2-isopropylidene-α-L-threose involving carbon homologation and microwave-assisted Vorbrüggen coupling. These compounds were evaluated against a panel of viruses, cancer cell lines, adenosine receptors, thymidine kinases and thymidylate kinase of M. tuberculosis.

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Chicago
Toti, Kiran, Marco Derudas, Davy Sinnaeve, José Martins, Christopher McGuigan, Jan Balzarini, Kenneth A Jacobson, and Serge Van Calenbergh. 2012. “Synthesis and Biological Evaluation of Apionucleosides and Their Protides.” In Nucleosides, Nucleotides and Nucleic Acids, 20th International Roundtable, Abstracts, 51–51. International Society of Nucleosides, Nucleotides and Nucleic Acids (IS3NA).
APA
Toti, K., Derudas, M., Sinnaeve, D., Martins, J., McGuigan, C., Balzarini, J., Jacobson, K. A., et al. (2012). Synthesis and biological evaluation of apionucleosides and their protides. Nucleosides, Nucleotides and Nucleic Acids, 20th International roundtable, Abstracts (pp. 51–51). Presented at the 20th International roundtable on Nucleosides, Nucleotides and Nucleic Acids, International Society of Nucleosides, Nucleotides and Nucleic Acids (IS3NA).
Vancouver
1.
Toti K, Derudas M, Sinnaeve D, Martins J, McGuigan C, Balzarini J, et al. Synthesis and biological evaluation of apionucleosides and their protides. Nucleosides, Nucleotides and Nucleic Acids, 20th International roundtable, Abstracts. International Society of Nucleosides, Nucleotides and Nucleic Acids (IS3NA); 2012. p. 51–51.
MLA
Toti, Kiran, Marco Derudas, Davy Sinnaeve, et al. “Synthesis and Biological Evaluation of Apionucleosides and Their Protides.” Nucleosides, Nucleotides and Nucleic Acids, 20th International Roundtable, Abstracts. International Society of Nucleosides, Nucleotides and Nucleic Acids (IS3NA), 2012. 51–51. Print.
@inproceedings{2984014,
  abstract     = {We report the synthesis of the A and T 2',3'-dideoxyapionucleosides and their corresponding Pro-Tide derivatives from 1,2-isopropylidene-\ensuremath{\alpha}-L-threose involving carbon homologation and microwave-assisted Vorbr{\"u}ggen coupling. These compounds were evaluated against a panel of viruses, cancer cell lines, adenosine receptors, thymidine kinases and thymidylate kinase of M. tuberculosis.},
  author       = {Toti, Kiran and Derudas, Marco and Sinnaeve, Davy and Martins, Jos{\'e} and McGuigan, Christopher and Balzarini, Jan and Jacobson, Kenneth A and Van Calenbergh, Serge},
  booktitle    = {Nucleosides, Nucleotides and Nucleic Acids, 20th International roundtable, Abstracts},
  language     = {eng},
  location     = {Montr{\'e}al, QU, Canada},
  pages        = {51--51},
  publisher    = {International Society of Nucleosides, Nucleotides and Nucleic Acids (IS3NA)},
  title        = {Synthesis and biological evaluation of apionucleosides and their protides},
  year         = {2012},
}