Romain Merceron

Structure-aided optimization of non-nucleoside M. tuberculosis thymidylate kinase inhibitors

Lijun Song (UGent) , Romain Merceron (UGent) , Fabian Hulpia (UGent) , Ainhoa Lucia, Begona Gracia, Yanlin Jian (UGent) , Martijn Risseeuw (UGent) , Toon Verstraelen (UGent) , Paul Cos, Jose A. Ainsa, et al.

(2021) EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. 225.

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Distinct EH domains of the endocytic TPLATE complex confer lipid and protein binding

Klaas Yperman (UGent) , Anna Papageorgiou, Romain Merceron (UGent) , Steven De Munck (UGent) , Yehudi Bloch (UGent) , Dominique Eeckhout (UGent) , Qihang Jiang (UGent) , Pieter Tack (UGent) , Rosa Grigoryan (UGent) , Thomas Evangelidis, et al.

(2021) NATURE COMMUNICATIONS. 12(1).

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Molecular architecture of the endocytic TPLATE complex

Klaas Yperman (UGent) , Jie Wang (UGent) , Dominique Eeckhout (UGent) , Joanna Winkler (UGent) , Lam Dai Vu (UGent) , Michaël Vandorpe (UGent) , Peter Grones (UGent) , Evelien Mylle (UGent) , Michael Kraus (UGent) , Romain Merceron (UGent) , et al.

(2021) SCIENCE ADVANCES. 7(9).

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Endeavors towards transformation of M. tuberculosis thymidylate kinase (MtbTMPK) inhibitors into potential antimycobacterial agents

Yanlin Jian (UGent) , Romain Merceron (UGent) , Steven De Munck (UGent) , He Eun Forbes, Fabian Hulpia (UGent) , Martijn Risseeuw (UGent) , Kristof Van Hecke (UGent) , Savvas Savvides (UGent) , Hélène Munier-Lehmann, Helena I. M. Boshoff, et al.

(2020) EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY. 206.

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Structural basis of latent TGF-β1 presentation and activation by GARP on human regulatory T cells

Stephanie Lienart, Romain Merceron (UGent) , Christophe Vanderaa, Fanny Lambert, Didier Colau, Julie Stockis, Bas van der Woning, Hans De Haard, Michael Saunders, Pierre G Coulie, et al.

(2018) SCIENCE. 362(6417). p.952-956

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Structure guided lead generation toward nonchiral M. tuberculosis thymidylate kinase inhibitors

Lijun Song (UGent) , Romain Merceron (UGent) , Begoña Gracia, Ainhoa Lucía Quintana, Martijn Risseeuw (UGent) , Fabian Hulpia (UGent) , Paul Cos, José A Aínsa, Hélène Munier-Lehmann, Savvas Savvides (UGent) , et al.

(2018) JOURNAL OF MEDICINAL CHEMISTRY. 61(7). p.2753-2775

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Structural activation of pro-inflammatory human cytokine IL-23 by cognate IL-23 receptor enables recruitment of the shared receptor IL-12Rβ1

Yehudi Bloch (UGent) , Laura Bouchareychas, Romain Merceron (UGent) , Katarzyna Skladanowska (UGent) , Lien Van den Bossche (UGent) , Sammy Detry (UGent) , Srinath Govindarajan (UGent) , Dirk Elewaut (UGent) , Filomeen Haerynck (UGent) , Melissa Dullaers (UGent) , et al.

(2018) IMMUNITY. 48(1). p.45-58

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The design and synthesis of inhibitors of Mycobacterium tuberculosis thymidylate kinase (MtTMPK)

Lijun Song (UGent) , Martijn Risseeuw (UGent) , Fabian Hulpia (UGent) , Romain Merceron (UGent) , Savvas Savvides (UGent) , Hélène Munier-Lehmann and Serge Van Calenbergh (UGent)

(2016) Nucleosides, Nucleotides and Nucleic Acids, XXII Round table, Abstracts. p.180-180

Academic Bibliography

Romain Merceron

Structure-aided optimization of non-nucleoside M. tuberculosis thymidylate kinase inhibitors

Distinct EH domains of the endocytic TPLATE complex confer lipid and protein binding

Molecular architecture of the endocytic TPLATE complex

Endeavors towards transformation of M. tuberculosis thymidylate kinase (MtbTMPK) inhibitors into potential antimycobacterial agents

Structural basis of latent TGF-β1 presentation and activation by GARP on human regulatory T cells

Structure guided lead generation toward nonchiral M. tuberculosis thymidylate kinase inhibitors

Structural activation of pro-inflammatory human cytokine IL-23 by cognate IL-23 receptor enables recruitment of the shared receptor IL-12Rβ1

The design and synthesis of inhibitors of Mycobacterium tuberculosis thymidylate kinase (MtTMPK)

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