Yves Depetter

Journal Article
A1
open access

Expedient synthesis of lupulones and their derivatization to 2,8-7H-dihydrochromen-7-ones

Lena Decuyper, Gurkirat Kaur, Charlotte Versyck, Eline Blondeel, Yves Depetter, Kristof Van Hecke (UGent) and Matthias D'hooghe (UGent)

(2020) CHEMISTRYOPEN. 9(4). p.442-444

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Journal Article
A1
open access

Synthesis of indoline‐based benzhydroxamic acids as potential HDAC6 inhibitors

Yves Depetter, Silke Geurs (UGent) , Jorick Franceus (UGent) , Damijan Knez, Tom Desmet (UGent) , Karolien De Bosscher (UGent) , Olivier De Wever (UGent) , Stanislav Gobec and Matthias D'hooghe (UGent)

(2019) CHEMISTRYSELECT. 4(42). p.12308-12312

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Selective pharmacological inhibitors of HDAC6 reveal biochemical activity but functional tolerance in cancer models

Yves Depetter, Silke Geurs (UGent) , Rob De Vreese (UGent) , Sophie Goethals, Elien Vandoorn (UGent) , Alien Laevens, Jonas Steenbrugge (UGent) , Evelyne Meyer (UGent) , Pascal de Tullio, Marc Bracke (UGent) , et al.

(2019) INTERNATIONAL JOURNAL OF CANCER. 145(3). p.735-747

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PhD Thesis
open access

Synthesis of selective HDAC6 inhibitors and their evaluation in cancer models

Yves Depetter

(2019)

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Assessment of the trifluoromethyl ketone functionality as an alternative zinc-binding group for selective HDAC6 inhibition

Yves Depetter, Silke Geurs (UGent) , Flore Vanden Bussche, Rob De Vreese (UGent) , Jorick Franceus (UGent) , Tom Desmet (UGent) , Olivier De Wever (UGent) and Matthias D'hooghe (UGent)

(2018) MEDCHEMCOMM. 9(6). p.1011-1016

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Synthesis of potent and selective HDAC6 inhibitors bearing a cyclohexane- or cycloheptane-annulated 1,5-benzothiazepine scaffold

Rob De Vreese (UGent) , Lisa Galle, Yves Depetter, Jorick Franceus (UGent) , Tom Desmet (UGent) , Kristof Van Hecke (UGent) , Veronick Benoy, Ludo Van Den Bosch and Matthias D'hooghe (UGent)

(2017) CHEMISTRY-A EUROPEAN JOURNAL. 23(1). p.128-136

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Synthesis and SAR assessment of novel Tubathian analogs in the pursuit of potent and selective HDAC6 inhibitors

Rob De Vreese (UGent) , Yves Depetter, Tom Verhaeghe (UGent) , Tom Desmet (UGent) , Veronick Benoy, Wanda Haeck, Ludo Van Den Bosch and Matthias D'hooghe (UGent)

(2016) ORGANIC & BIOMOLECULAR CHEMISTRY. 14(8). p.2537-2549

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Synthesis and anticancer properties of new (dihydro)pyranonaphthoquinones and their epoxy analogs

Anh Dang Thi Tuyet, Ha Vu Thi Thu, Thi Phuong Hoang, Ha Nguyen Thanh, Pham The Chinh, Vu Duc Cuong, Yves Depetter, Van Nguyen Tuyen and Matthias D'hooghe (UGent)

(2015) BIOORGANIC & MEDICINAL CHEMISTRY LETTERS. 25(16). p.3355-3358

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Expedient stereoselective synthesis of new dihydropyrano- and dihydrofuranonaphthoquinones

Tuyet Anh Dang Thi, Yves Depetter, Karen Mollet (UGent) , Hoang Thi Phuong, Doan Vu Ngoc, Chinh Pham The, Ha Thanh Nguyen, Thu Ha Nguyen Thi, Hung Huy Nguyen, Matthias D'hooghe (UGent) , et al.

(2015) TETRAHEDRON LETTERS. 56(19). p.2422-2425

Academic Bibliography

Yves Depetter

Expedient synthesis of lupulones and their derivatization to 2,8-7H-dihydrochromen-7-ones

Synthesis of indoline‐based benzhydroxamic acids as potential HDAC6 inhibitors

Selective pharmacological inhibitors of HDAC6 reveal biochemical activity but functional tolerance in cancer models

Synthesis of selective HDAC6 inhibitors and their evaluation in cancer models

Assessment of the trifluoromethyl ketone functionality as an alternative zinc-binding group for selective HDAC6 inhibition

Synthesis of potent and selective HDAC6 inhibitors bearing a cyclohexane- or cycloheptane-annulated 1,5-benzothiazepine scaffold

Synthesis and SAR assessment of novel Tubathian analogs in the pursuit of potent and selective HDAC6 inhibitors

Synthesis and anticancer properties of new (dihydro)pyranonaphthoquinones and their epoxy analogs

Expedient stereoselective synthesis of new dihydropyrano- and dihydrofuranonaphthoquinones

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