dr. apr. Fabian Hulpia
No current affiliation with UGent
- ORCID iD
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0000-0002-7470-3484
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- Journal Article
- A1
- open access
Phenotypic evaluation of nucleoside analogues against Trypanosoma cruzi infection : in vitro and in vivo approaches
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- Journal Article
- A1
- open access
Exploration of 6-methyl-7-(hetero)aryl-7-deazapurine ribonucleosides as antileishmanial agents
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- Journal Article
- A1
- open access
Nucleoside analogues for the treatment of animal trypanosomiasis
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- Journal Article
- A1
- open access
A Toxoplasma gondii oxopurine transporter binds nucleobases and nucleosides using different binding modes
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- Journal Article
- A1
- open access
Ex vivo feedback control of neurotransmission using a photocaged adenosine A1 receptor agonist
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Phenethyl-4-ANPP : a marginally active byproduct suggesting a switch in illicit fentanyl synthesis routes
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- Journal Article
- A2
- open access
7-Aryl-7-deazapurine 3 '-deoxyribonucleoside derivative as a novel lead for Chagas' disease therapy : in vitro and in vivo pharmacology
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- Journal Article
- A1
- open access
6-Methyl-7-deazapurine nucleoside analogues as broad-spectrum antikinetoplastid agents
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- Journal Article
- A1
- open access
Deazapurine nucleoside analogues for the treatment of Trichomonas vaginalis
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Structure-aided optimization of non-nucleoside M. tuberculosis thymidylate kinase inhibitors
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- Conference Paper
- C3
- open access
Optical control of excitatory transmission in hippocampal slices with photoactive adenosine A1 receptor agonist
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- Conference Paper
- C3
- open access
Optical control of excitatory transmission in hippocampal slices with photoactive adenosine A1 receptor agonist
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- Journal Article
- A1
- open access
4E interacting protein as a potential novel drug target for nucleoside analogues in Trypanosoma brucei
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- Journal Article
- A1
- open access
Synthesis and evaluation of 3′-fluorinated 7-deazapurine nucleosides as antikinetoplastid agents
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6‐methyl‐7‐aryl‐7‐deazapurine nucleosides as anti‐trypanosoma cruzi agents : structure‐activity relationship and in vivo efficacy
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2-((3,5-Dinitrobenzyl)thio)quinazolinones : potent antimycobacterial agents activated by deazaflavin (F420)-dependent nitroreductase (Ddn)
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- Journal Article
- A1
- open access
Report on a new opioid NPS : chemical and in vitro functional characterization of a structural isomer of the MT-45 derivative diphenpipenol
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- Miscellaneous
- open access
Positively selected modifications in the pore of TbAQP2 allow pentamidine to enter Trypanosoma brucei
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- Journal Article
- A1
- open access
Positively selected modifications in the pore of TbAQP2 allow pentamidine to enter Trypanosoma brucei
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- Journal Article
- A1
- open access
First report on brorphine : the next opioid on the deadly new psychoactive substance horizon?
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- Journal Article
- A1
- open access
Endeavors towards transformation of M. tuberculosis thymidylate kinase (MtbTMPK) inhibitors into potential antimycobacterial agents
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- Journal Article
- A1
- open access
1-(1-Arylethylpiperidin-4-yl)thymine analogs as antimycobacterial TMPK inhibitors
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- Journal Article
- A1
- open access
Structure-activity relationship exploration of 3’-deoxy-7-deazapurine nucleoside analogues as anti-Trypanosoma brucei agents
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Synthesis and structure activity relationships of cyanopyridone based anti-tuberculosis agents
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3'-Deoxyribofuranosyl 7-deazapurine nucleoside analogues : a new class of highly potent antitrypanosomal agents
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Deazapurine nucleoside analogues as potent anti-Trypanosoma cruzi agents
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- Journal Article
- A1
- open access
6-O-alkylated 7-deazainosine nucleoside analogues : discovery of potent and selective anti-sleeping sickness agents
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Report on a novel emerging class of highly potent benzimidazole NPS opioids : chemical and in vitro functional characterization of isotonitazene
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Design and synthesis of trypanocidal purine nucleoside analogues : discovery of lead compounds for the treatment of sleeping sickness
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- Journal Article
- A1
- open access
Combining tubercidin and cordycepin scaffolds results in highly active candidates to treat late-stage sleeping sickness
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Purine nucleoside analogs as highly potent leads for the treatment of human African trypanosomiasis
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Novel pyrazolo[3,4-d]pyrimidine nucleosides : promising hits for Chagas disease and Leishmaniasis
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Synthesis and evaluation of 3’-deoxy-3’-fluoro-7-deazapurine nucleosides as antikinetoplastid agents
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Purine nucleoside analogs as highly potent leads for the treatment of human African trypanosomiasis
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Discovery of 7-aryl-7-deazapurine 3'-deoxyribofuranosyl nucleoside analogues as anti-Trypanosoma cruzi agents
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Discovery of pyrrolo[2,3-b]pyridine (1,7-dideazapurine) nucleoside analogues as anti-Trypanosoma cruzi agents
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3’-Deoxy-3’-fluoro-7-deazapurine nucleosides : synthesis and evaluation against kinetoplastid parasites
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Discovery of pyrrolo[2,3-b]pyridine nucleoside analogues as anti-Trypanosoma cruzi agents
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- Journal Article
- A1
- open access
New fluoroethyl phenylalanine analogues as potential LAT1-targeting PET tracers for glioblastoma
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Revisiting tubercidin against kinetoplastid parasites : aromatic substitutions at position 7 improve activity and reduce toxicity
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C7 substituted 7-deaza adenosines : design and synthesis of nucleosides with potent antitrypanosomal activity
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Discovery of novel 7-aryl 7-deazapurine 3'-deoxy-ribofuranosyl nucleosides with potent activity against Trypanosoma cruzi
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- Journal Article
- A1
- open access
Synthesis of a 3'-C-ethynyl-β-D-ribofuranose purine nucleoside library : discovery of C7-deazapurine analogs as potent antiproliferative nucleosides
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Design and synthesis of a purine nucleoside library : phenotypic discovery of antikinetoplastid agents
(2018) -
Structure guided lead generation toward nonchiral M. tuberculosis thymidylate kinase inhibitors
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Novel 3'-deoxy purine nucleoside analogs as highly potent leads for human African trypanosomiasis
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The design and synthesis of inhibitors of Mycobacterium tuberculosis thymidylate kinase (MtTMPK)
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Purine-mimicking 3'-ethynylribofuranose nucleosides: new opportunities for an old sugar modification
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Purine-mimicking 3’-ethynylribofuranose nucleosides : new opportunities for an old sugar modification
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C-3’-ethynylnucleosides: an old modification going viral
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Exploring the purine core of 3'-C-ethynyladenosine (EAdo) in search of novel nucleoside therapeutics
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Synthesis, in vitro and in vivo small-animal SPECT evaluation of novel technetium labeled bile acid analogues to study (altered) hepatic transporter function
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- Conference Paper
- C3
- open access
The design and synthesis of inhibitors of Mycobacterium tuberculosis thymidylate kinase (MtTMPK)
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Novel nucleoside therapeutics :'Min(d)ing the gap'
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- Conference Paper
- C3
- open access
Phenotypic screening of a focused nucleoside library
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- Conference Paper
- C3
- open access
In search of novel nucleoside therapeutics: exploring the purine core of 3'-C-ethynyladenosine
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- Conference Paper
- C3
- open access
The design and synthesis of inhibitors of Mycobacterium tuberculosis thymidylate kinase (MtTMPK)