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Selective pharmacological inhibitors of HDAC6 reveal biochemical activity but functional tolerance in cancer models
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Assessment of the trifluoromethyl ketone functionality as an alternative zinc-binding group for selective HDAC6 inhibition
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- Journal Article
- A1
- open access
Synthesis and applications of benzohydroxamic acid-based histone deacetylase inhibitors
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- Journal Article
- A1
- open access
Exploration of thiaheterocyclic hHDAC6 inhibitors as potential antiplasmodial agents
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Synthesis of bis-8-hydroxyquinolines via an imination or a Suzuki-Miyaura coupling approach
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- PhD Thesis
- open access
Synthesis of thiaheterocyclic benzohydroxamic acids and evaluation of their HDAC6 inhibitory activity
(2017) -
- Journal Article
- A1
- open access
Synthesis of potent and selective HDAC6 inhibitors bearing a cyclohexane- or cycloheptane-annulated 1,5-benzothiazepine scaffold
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- Journal Article
- A1
- open access
Synthesis and SAR assessment of novel Tubathian analogs in the pursuit of potent and selective HDAC6 inhibitors
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Converting bulk sugars into prebiotics : semirational design of a transglucosylase with controlled selectivity
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Synthesis and biological assessment of novel N-(hydroxy/methoxy)alkyl β-enaminone curcuminoids
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Synthesis of novel curcuminoids accommodating a central β-enaminone motif and their impact on cell growth and oxidative stress
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Synthesis of novel thymine-β-lactam hybrids and evaluation of their anti-tumor activity
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Synthesis of benzothiophene-based hydroxamic acids as potent and selective HDAC6 inhibitors
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Synthesis of novel thymine-β-lactam hybrids and evaluation of their anti-tumor activity
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Synthesis of novel thymine-β-lactam hybrids and evaluation of their anti-tumor activity
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Engineering the specificity of trehalose phosphorylase as a general strategy for the production of glycosyl phosphates
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Potent and selective HDAC6 inhibitory activity of N-(4-hydroxycarbamoylbenzyl)-1,2,4,9-tetrahydro-3-thia-9-azafluorenes as novel sulfur analogues of Tubastatin A
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Design, synthesis and antiviral evaluation of purine-β-lactam and purine-aminopropanol hybrids
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- Journal Article
- A1
- open access
N-Heterocyclic carbene/Brønsted acid cooperative catalysis as a powerful tool in organic synthesis