Ghent University Academic Bibliography

Journal Article
A1
open access

Off-target activity of NBOMes and NBOMe analogs at the mu opioid receptor

Marie Deventer (UGent) , Mattias Persson, Antonio Laus, Eline Pottie (UGent) , Annelies Cannaert (UGent) , Graziella Tocco, Henrik Green and Christophe Stove (UGent)

(2023) ARCHIVES OF TOXICOLOGY. 97(5). p.1367-1384

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Machine learning to assist in large-scale, activity-based synthetic cannabinoid receptor agonist screening of serum samples

Liesl Janssens (UGent) , Dimitri Boeckaerts (UGent) , Simon Hudson, Daria Morozova, Annelies Cannaert (UGent) , David M. Wood, Caitlin Wolfe, Bernard De Baets (UGent) , Michiel Stock (UGent) , Paul, I Dargan, et al.

(2022) CLINICAL CHEMISTRY. 68(7). p.906-916

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Journal Article
A1
open access

Are the N-demethylated metabolites of U-47700 more active than their parent compound? In vitro mu-opioid receptor activation of N-desmethyl-U-47700 and N,N-bisdesmethyl-U-47700

Frederike Nordmeier, Annelies Cannaert (UGent) , Christophe Stove (UGent) , Peter H. Schmidt, Markus R. Meyer and Nadine Schaefer

(2022) DRUG TESTING AND ANALYSIS. 14(4). p.713-717

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NNL-3 : a synthetic intermediate or a new class of hydroxybenzotriazole esters with cannabinoid receptor activity?

Adam Ametovski, Elizabeth A. Cairns, Katharina Elisabeth Grafinger, Annelies Cannaert (UGent) , Marie Deventer (UGent) , Shuli Chen, Xinyi Wu, Caitlin E. Shepperson, Felcia Lai, Ross Ellison, et al.

(2021) ACS CHEMICAL NEUROSCIENCE. 12(21). p.4020-4036

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Systematic evaluation of a panel of 30 synthetic cannabinoid receptor agonists structurally related to MMB-4en-PICA, MDMB-4en-PINACA, ADB-4en-PINACA, and MMB-4CN-BUTINACA using a combination of binding and different CB1 receptor activation assays-Part II: Structure activity relationship assessment via a beta-arrestin recruitment assay

Katharina Grafinger, Annelies Cannaert (UGent) , Adam Ametovski, Eric Sparkes, Elizabeth Cairns, Samuel D. Banister, Volker Auwarter and Christophe Stove (UGent)

(2021) DRUG TESTING AND ANALYSIS. 13(7). p.1402-1411

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Systematic evaluation of a panel of 30 synthetic cannabinoid receptor agonists structurally related to MMB-4en-PICA, MDMB-4en-PINACA, ADB-4en-PINACA, and MMB-4CN-BUTINACA using a combination of binding and different CB1 receptor activation assays: Part I-Synthesis, analytical characterization, and binding affinity for human CB1 receptors

Edward Pike, Katharina Grafinger, Annelies Cannaert (UGent) , Adam Ametovski, Jia Lin Luo, Eric Sparkes, Elizabeth A. Cairns, Ross Ellison, Roy Gerona, Christophe Stove (UGent) , et al.

(2021) DRUG TESTING AND ANALYSIS. 13(7). p.1383-1401

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Journal Article
A1
open access

Systematic evaluation of a panel of 30 synthetic cannabinoid receptor agonists structurally related to MMB-4en-PICA, MDMB-4en-PINACA, ADB-4en-PINACA, and MMB-4CN-BUTINACA using a combination of binding and different CB1 receptor activation assays : part III : The G protein pathway and critical comparison of different assays

Katharina Elisabeth Grafinger, Marthe Vandeputte (UGent) , Annelies Cannaert (UGent) , Adam Ametovski, Eric Sparkes, Elizabeth Cairns, Patrick Osamu Juchli, Belal Haschimi, Benedikt Pulver, Samuel D. Banister, et al.

(2021) DRUG TESTING AND ANALYSIS. 13(7). p.1412-1429

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The next generation of synthetic cannabinoids : detection, activity, and potential toxicity of pent-4en and but-3en analogues including MDMB-4en-PINACA

Alex J. Krotulski, Annelies Cannaert (UGent) , Christophe Stove (UGent) and Barry K. Logan

(2021) DRUG TESTING AND ANALYSIS. 13(2). p.427-438

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Diagnosing intake and rationalizing toxicities associated with 5F-MDMB-PINACA and 4F-MDMB-BINACA abuse

Wen Lie, Eleanor Jing Yi Cheong, Evelyn Mei Ling Goh, Hooi Yan Moy, Annelies Cannaert (UGent) , Christophe Stove (UGent) and Eric Chun Yong Chan

(2021) ARCHIVES OF TOXICOLOGY. 95(2). p.489-508

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Shape matters : the application of activity-based in vitro bioassays and chiral profiling to the pharmacological evaluation of synthetic cannabinoid receptor agonists in drug-infused papers seized in prisons

Lysbeth H. Antonides, Annelies Cannaert (UGent) , Caitlyn Norman, Niamh NicDaeid, Oliver B. Sutcliffe, Christophe Stove (UGent) and Craig McKenzie

(2021) DRUG TESTING AND ANALYSIS. 13(3). p.628-643

Academic Bibliography

Off-target activity of NBOMes and NBOMe analogs at the mu opioid receptor

Machine learning to assist in large-scale, activity-based synthetic cannabinoid receptor agonist screening of serum samples

Are the N-demethylated metabolites of U-47700 more active than their parent compound? In vitro mu-opioid receptor activation of N-desmethyl-U-47700 and N,N-bisdesmethyl-U-47700

NNL-3 : a synthetic intermediate or a new class of hydroxybenzotriazole esters with cannabinoid receptor activity?

The next generation of synthetic cannabinoids : detection, activity, and potential toxicity of pent-4en and but-3en analogues including MDMB-4en-PINACA

Diagnosing intake and rationalizing toxicities associated with 5F-MDMB-PINACA and 4F-MDMB-BINACA abuse

Shape matters : the application of activity-based in vitro bioassays and chiral profiling to the pharmacological evaluation of synthetic cannabinoid receptor agonists in drug-infused papers seized in prisons

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